Design, Synthesis and Biological Evaluation of 1-Ethyl-3-(thiazol-2-yl)urea Derivatives as Escherichia coli DNA Gyrase Inhibitors

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Tomašič , T , Barančoková , M , Zidar , N , Ilaš , J , Tammela , P S M & Kikelj , D 2018 , ' Design, Synthesis and Biological Evaluation of 1-Ethyl-3-(thiazol-2-yl)urea Derivatives as Escherichia coli DNA Gyrase Inhibitors ' , Archiv der Pharmazie : Chemistry in life sciences , vol. 351 , no. 1 , e1700333 . https://doi.org/10.1002/ardp.201700333

Title: Design, Synthesis and Biological Evaluation of 1-Ethyl-3-(thiazol-2-yl)urea Derivatives as Escherichia coli DNA Gyrase Inhibitors
Author: Tomašič, Tihomir; Barančoková, Michaela; Zidar, Nace; Ilaš, Janez; Tammela, Päivi Sirpa Marjaana; Kikelj, Danijel
Contributor: University of Helsinki, Faculty of Pharmacy
Date: 2018-01-03
Language: eng
Number of pages: 16
Belongs to series: Archiv der Pharmazie : Chemistry in life sciences
ISSN: 0365-6233
URI: http://hdl.handle.net/10138/237145
Subject: 317 Pharmacy
Antibacterial
DNA gyrase
Ethylurea
INHIBITOR
THIAZOLE
antibacterial
DNA gyrase
ethylurea
inhibitor
thiazole
STRUCTURE-GUIDED DESIGN
ATP-BINDING-SITE
TOPOISOMERASE-IV
ANTIBACTERIAL ACTIVITY
B INHIBITORS
N-PHENYLINDOLAMIDES
IIA TOPOISOMERASES
DISCOVERY
POTENT
AGENTS
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